NSTK · 01.2026Independent supplement reference
NutriStack
Edition 1.0Reviewed May 26, 2026

Supplement·Interactions·Reviewed June 9, 2026

L-Citrulline interactions.

L-Citrulline has 32 documented interactions in the NutriStack database: 1 to avoid or watch closely, 22 that need timing or caution, and 9 that work synergistically. The full list, with what each pairing does, is below.

In short

L-Citrulline at a glance.

A quick, data-grounded summary. The full table is below.

L-Citrulline has 32 documented interactions in the NutriStack database: 1 to avoid or watch closely, 22 that need timing or caution, and 9 that work synergistically. The full list, with what each pairing does, is below.

Interactions

Everything that interacts with l-citrulline.

Every supplement and medication in the NutriStack database with a documented interaction with this substance, highest-severity first. Open any pair for the mechanism and sources.

SubstanceInteractionWhat happens
Citrulline MalateConflictCitrulline malate already supplies citrulline, so adding L-citrulline can create duplicate high dosing and GI effects.
Agmatine SulfateCautionBoth affect nitric oxide or vascular pathways, but agmatine may modulate nitric oxide synthase unpredictably.
AlfuzosinCautionL-Citrulline increases systemic arginine availability and can modestly lower blood pressure. Alfuzosin can also contribute to blood-pressure... details →
AmlodipineCautionL-Citrulline is converted to L-arginine and raises plasma arginine more efficiently than oral arginine itself, producing nitric-oxide-mediated... details →
CandesartanCautionL-Citrulline may add to the blood-pressure-lowering effect of Candesartan.
CaptoprilCautionL-Citrulline may add to the blood-pressure-lowering effect of Captopril.
ChlorthalidoneCautionL-Citrulline can modestly lower blood pressure through the arginine-nitric oxide pathway. Chlorthalidone has sustained antihypertensive and diuretic... details →
D-Aspartic AcidCautionL-Citrulline is one of the most common nitric oxide boosters in pre-workout and pump products, and it reliably elevates plasma arginine and nitric...
FelodipineCautionL-Citrulline may add to the blood-pressure-lowering effect of Felodipine.
HydrochlorothiazideCautionL-Citrulline can increase arginine availability and modestly lower systolic blood pressure. Hydrochlorothiazide also lowers blood pressure, so the... details →
Isosorbide MononitrateCautionL-citrulline increases L-arginine availability and can lower blood pressure through nitric oxide pathways. Isosorbide mononitrate is an organic... details →
LabetalolCautionL-Citrulline may add to the blood-pressure-lowering effect of Labetalol.
MetoprololCautionL-Citrulline is converted to L-arginine and raises plasma arginine more efficiently than arginine itself, producing nitric-oxide-mediated... details →
NebivololCautionL-Citrulline may add to the blood-pressure-lowering effect of Nebivolol.
NitroglycerinCautionL-citrulline raises circulating L-arginine and can support nitric-oxide-mediated blood pressure lowering. Nitroglycerin also works through nitric... details →
Pentadeca Arginate (PDA)CautionPDA is marketed as an arginate salt and related BPC-157 animal data involve nitric oxide pathways; L-citrulline can raise nitric oxide availability.
PerindoprilCautionL-Citrulline may add to the blood-pressure-lowering effect of Perindopril.
QuinaprilCautionL-Citrulline may add to the blood-pressure-lowering effect of Quinapril.
SilodosinCautionL-citrulline can increase nitric oxide availability and may add to silodosin-related dizziness or orthostatic hypotension.
TamsulosinCautionL-Citrulline raises plasma arginine and can lower blood pressure through nitric-oxide-mediated vasodilation. Tamsulosin has a documented association... details →
TelmisartanCautionL-Citrulline may add to the blood-pressure-lowering effect of Telmisartan.
Timolol OphthalmicCautionL-Citrulline increases arginine availability and can modestly lower blood pressure. Timolol eye drops can reach systemic circulation and produce... details →
VIP (Vasoactive Intestinal Peptide)CautionL-citrulline can increase nitric oxide-mediated vasodilation and may add to VIP-related flushing or low blood pressure.
Beetroot Extract (Dietary Nitrate)SynergyBoth increase nitric oxide availability and may additively lower blood pressure.
Beta-AlanineSynergyBeta-alanine and L-citrulline are frequently combined and may give complementary gains in high-intensity and endurance performance.
L-ArginineSynergyCitrulline is converted to arginine in the kidney, raising plasma arginine higher and longer than oral arginine alone. Combined use provides...
LisinoprilSynergyL-Citrulline is converted to arginine in the kidney and produces sustained increases in nitric oxide. A meta-analysis of clinical trials reported... details →
Oligonol (Lychee Polyphenol)SynergyL-Citrulline raises plasma arginine and nitric oxide production while Oligonol supports endothelial function and microcirculation; combined use may...
Pine Bark ExtractSynergyL-citrulline raises plasma arginine and nitric oxide production, complementing pine bark extract's enhancement and protection of endothelial nitric...
SildenafilSynergyL-Citrulline can increase L-arginine availability and nitric-oxide-dependent signaling, which is upstream of sildenafil's PDE5 effect. In a small...
TadalafilSynergyL-Citrulline can raise plasma L-arginine and nitric-oxide signaling, while tadalafil preserves cGMP by inhibiting PDE5. A small randomized crossover...
TaurineSynergyBoth amino acids support endothelial function and exercise performance, and are commonly combined for complementary vascular and ergogenic effects.
Go deeper

The full l-citrulline profile.

Benefits, dosing by goal, forms, and the cited evidence for this supplement.

FAQ

Common l-citrulline questions.

Quick answers drawn from the table above.

What interacts with L-Citrulline?

In the NutriStack database, L-Citrulline has 32 documented interactions with other supplements and medications. The most notable include Citrulline Malate, Agmatine Sulfate, Alfuzosin, Amlodipine, and Candesartan.

What should you not take with L-Citrulline?

L-Citrulline is flagged against 1 substance in the database, including Citrulline Malate. Review these with a clinician before combining, especially alongside prescription medications.

What works well with L-Citrulline?

L-Citrulline pairs synergistically with Beetroot Extract (Dietary Nitrate), Beta-Alanine, L-Arginine, Lisinopril, and Oligonol (Lychee Polyphenol) in the NutriStack database. Synergy still depends on dose and timing; open any pair for the detail.

Can you take L-Citrulline with Citrulline Malate?

NutriStack classifies the L-Citrulline and Citrulline Malate pairing as conflict: Citrulline malate already supplies citrulline, so adding L-citrulline can create duplicate high dosing and GI effects. Count total citrulline from all products and reduce doses if stacking.

Check your whole stack

See how l-citrulline fits your routine.

NutriStack screens your full stack for interactions and timing conflicts, and updates the moment you change it.

NutriStack is an informational and organizational tool, not a medical service, and not a substitute for professional advice. Always consult a qualified healthcare professional before starting, stopping, or changing any supplement or medication.